Bretazenil Powder

Bretazenil is a benzodiazepine analog known for its unique action as a partial agonist at GABA-A receptors. Unlike full benzodiazepine agonists (e.g., diazepam), Bretazenil has a subtler profile, offering anxiolytic and anticonvulsant activity with reduced sedative and muscle relaxant effects.

Researchers utilize Bretazenil to investigate the role of GABA-A receptor subtypes, benzodiazepine tolerance, and the modulation of inhibitory neurotransmission. Due to its partial agonism, It is also of interest in exploring the mechanisms behind dependence, withdrawal, and receptor desensitization.

Dopechem.com provides high-purity Bretazenil powder for licensed laboratory, forensic, and analytical research. This compound is not intended for human or veterinary use.

🔬 Common Research Applications 

• GABA-A receptor modulation studies

• Investigating benzodiazepine tolerance and dependence

• CNS inhibitory signaling research

• Anticonvulsant mechanism analysis

• Receptor binding assays in neuropharmacology

⚠️ Potential Side Effects of Bretazenil Powder (in non-clinical models or misuse)

• Mild sedation at high concentrations

• Reduced locomotor activity

• Temporary anxiety or agitation in sensitive models

• Potential withdrawal symptoms upon cessation

• Muscle coordination impairment in test subjects

📦 Storage & Handling

• Store at -20°C in a dry, dark, and airtight container

• Use appropriate safety measures and PPE when handling